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HETEROCYCLIC COMPOUNDS AS HDAC INHIBITORS

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专利名称:HETEROCYCLIC COMPOUNDS AS HDAC

INHIBITORS

发明人:BALASUBRAMANIAN,

GOPALAN,RAJAGOPAL,SRIDHARAN,RATHINASAMY,SURESH,KILAMBI,

NARASIMHAN,RAJENDRAN,PRAVEEN,NARAYANAN, SHRIDHAR

申请号:IB2009007707申请日:20091210

公开号:WO2010073078A3公开日:20101104

摘要:The present invention relates to heterocyclic compounds of the generalformula (I) their derivatives, analogs, tautomeric forms, stereoisomers, geometricalisomers, polymorphs, hydrates, solvates, metabolites, prodrugs, pharmaceuticallyacceptable salts and compositions thereof. Also included is method for treatment ofproliferative conditions and cancer, conditions mediated by HDAC, in a mammalcomprising administering an effective amount of compound formula (I) as describedabove.

申请人:ORCHID RESEARCH LABORATORIES LTD.,BALASUBRAMANIAN,GOPALAN,RAJAGOPAL, SRIDHARAN,RATHINASAMY, SURESH,KILAMBI,NARASIMHAN,RAJENDRAN, PRAVEEN,NARAYANAN, SHRIDHAR

代理人:CHOPRA, Priyanka

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